Keto/enol epoxy steroids: a new structural class of HIV-1 Tat inhibitors

J Med Chem. 1993 Sep 3;36(18):2701-2. doi: 10.1021/jm00070a014.
No abstract available

MeSH terms

  • Androstanols / chemistry
  • Androstanols / pharmacology*
  • Androstenediols / chemistry
  • Androstenediols / pharmacology*
  • Cell Line
  • Gene Products, tat / antagonists & inhibitors*
  • Genes, tat
  • HIV-1 / chemistry*
  • Magnetic Resonance Spectroscopy
  • Molecular Structure
  • Transfection
  • tat Gene Products, Human Immunodeficiency Virus

Substances

  • Androstanols
  • Androstenediols
  • Gene Products, tat
  • tat Gene Products, Human Immunodeficiency Virus
  • 2-carbamoyl-4,5-epoxyandrost-2-ene-3,17-diol
  • 4,5-epoxy-17-hydroxy-2-methylsulfonyl-3-androstanone